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Synthesis and applications of the sulfur containing analogues of cyclic carbonates
Cyclic thiocarbonates are the sulfur containing analogues of the well-studied cyclic carbonates and are relatively poorly ...
Chiral sulfide and selenide catalysts for asymmetric halocyclizations and related reactions
Asymmetric organocatalysis using well-designed artificial chiral molecular catalysts is one of the most reliable methods t...
A Structure Activity Relationship Study of 3,4’-Dimethoxyflavone for ArlRS Inhibition in Staphylococcus aureus
Infections caused by methicillin-resistant Staphylococcus aureus (MRSA) are difficult to treat due to their resistance to ...
Kinetic resolution of sulfoxides with high enantioselectivity by a new homologue of methionine sulfoxide reductase B
Optically pure sulfoxides are noteworthy compounds that find wide applications in various industrial fields. Here we repor...
Copper-catalyzed radical-mediated intermolecular cyanomonofluoroalkylation of alkenes and alkynes
A novel copper-catalyzed three-component reaction of monofluoroalkylation agents, alkenes and TMSCN is described. In addit...
Deoxygenation of oximes for the synthesis of pyrrolines via hydroimination cyclization
Herein, we report the generation of iminyl radicals through photocatalytic deoxygenation of oximes with trivalent phosphin...
Hydrogen Bond Directed High Fidelity Optical Detection of Picric Acid: Single Driver through Diverse Road towards Same Destiny
High-fidelity optical detection of picric acid is the urge of the time due to its toxic and explosive nature. Moreover, Pi...
Synthesis, conformational stability and molecular structure of 4-aryl- and 4,5-diaryl-1,8-bis(dimethylamino)naphthalenes
4-Bromo- and 4,5-dibromo-1,8-bis(dimethylamino)naphthalenes were arylated with arylboronic acids under Suzuki reaction con...
Synthesis of Quinazolinones via Cp*Co(III)-Catalyzed C-H Functionalization of Primary Amides with Oxadiazolones
Multi-heteroatom heterocycle synthesis through direct C-H bond activation is methodologically appealing but synthetically ...
Catalytic Aminomethylative Etherification of N-Allenamides with N,O-Acetals Enabled by Lewis/Brønsted Acid Catalysis
A novel copper-catalyzed aminomethylative etherification of N-allenamides/ alkoxyallenes with N,O-acetals have been realiz...
Formal Synthesis of Cyclotheonellazole A
A convergent procedure for the formal synthesis of cyclotheonellazole A has been developed with high yields and excellent ...
Modular Synthesis of Fluorinated 2H-Thiophenes via [4+1] Cyclization of Enaminothiones
An efficient and straightforward synthetic method has been disclosed to construct trifluoromethyl 2H-thiophenes through [4...
Thia-Michael Addition: The Route to Promising Opportunities for Fast and Cysteine-Specific Modification
Over the last few decades, design and discovery of chemical reactions that enable modification of proteins at pre-determin...
Correction: An efficient metal free synthesis of 2-aminobenzothiozoles – a greener approach
Correction for ‘An efficient metal free synthesis of 2-aminobenzothiozoles – a greener approach’ by Krithika Ganesh et al....
Nickel-Catalysed Enantioselective Reaction of Secondary Phosphine Oxides and Activated Vinylcyclopropanes
Activated vinylcyclopropanes (VCPs) can form zwitterionic π-allylmetal species in the presence of transition metals and ar...
Stabilizing the hydroperoxyflavin intermediate formation via peptide appendage: A neutral flavoenzyme model
A bioinspired mimic for the stabilization of hydroperoxyflavin intermediate formation was designed and investigated for th...
Synthesis and Ring-Opening Metathesis Polymerisation of O-Alkoxy Benzothiadiazole Paracyclophane-1,9-dienes
Ortho-diethylhexyloxyphenylene benzothiadiazole paracyclophane-1,9-diene as a mixture of diastereomers was synthesized by ...
Factors influencing on-resin depsipeptide bond formation: Case studies on daptomycin- and brevicidine-derived sequences
Depsipeptides are an important class of bioactive natural products, where a growing number of genome-mined structures that...
Bimodal structural tuning of pyrrole-2-carboxamide-based transmembrane ion transport system
Pyrrole-2-carboxamide moiety is well known for its presence in various natural products and its use in anion receptor syst...