Gallic acid derived diarylpropanones exhibit synergistic antibacterial activities

WHO. Antimicrobial resistance. Key facts. 2023. https://www.who.int/news-room/fact-sheets/detail/antimicrobial-resistance.

Privalsky TM, Soohoo AM, Wang J, Walsh CT, Wright GD, Gordon EM, et al. Prospects for antibacterial discovery and development. J Am Chem Soc. 2021;143:21127–42.

Article  CAS  PubMed  PubMed Central  Google Scholar 

WHO. Global priority list of antibiotic-resistant bacteria to guide research, discovery, and development of new antibiotics. 2017. https://www.who.int/news/item/27-02-2017-who-publishes-list-of-bacteria-for-which-new-antibiotics-are-urgently-needed.

Murray CW, Rees DC. The rise of fragment-based drug discovery. Nat Chem. 2009;1:187–92.

Article  CAS  PubMed  Google Scholar 

Giordanetto F, Jin C, Willmore L, Feher M, Shaw DE. Fragment hits: what do they look like and how do they bind? J Med Chem. 2019;62:3381–94.

Article  CAS  PubMed  PubMed Central  Google Scholar 

Negi AS, Gautam Y, Alam S, Chanda D, Luqman S, Sarkar J, et al. Natural antitubulin agents: Importance of 3, 4, 5-trimethoxyphenyl fragment. Bioorg Med Chem. 2015;23:373–89.

Article  CAS  PubMed  Google Scholar 

Ustinov NB, Korshunoval AV, Gudimchuk NB. Protein complex NDC80: properties, functions, and possible role in pathophysiology of cell division. Biochemistry. 2020;85:448–62.

CAS  PubMed  Google Scholar 

Vos T, Allen C, Arora M, Barber RM, Bhutta ZA, et al. Global, regional, and national incidence, prevalence, and years lived with disability for 310 diseases and injuries, 1990–2015: a systematic analysis for the Global Burden of Disease Study 2015. The Lancet. 2016;388:1545–602.

Article  Google Scholar 

Zhang J, Gu Y, Chen B. Mechanisms of drug resistance in acute myeloid leukemia. Onco Targets Ther. 2019;12:1937–45.

Article  PubMed  PubMed Central  Google Scholar 

Hsu KS, Toda T. Ndc80 internal loop interacts with Dis1/TOG to ensure proper kinetochore-spindle attachment in fission yeast. Curr Biol. 2011;21:214–20.

Article  CAS  PubMed  PubMed Central  Google Scholar 

Field MC. The kinetochore and the origin of eukaryotic. Chromosome segregation. Proc Natl Acad Sci. 2019;116:12596–8.

Article  CAS  PubMed  PubMed Central  Google Scholar 

Anadón A, Martínez-Larrañaga MR, Ares I, Martínez MA. Biomarkers of drug toxicity and safety evaluation. In: Biomarkers in Toxicology. Chapter 38. 2nd ed. Academic Press, Elsevier Inc., USA; 2019. p. 655–91.

Hoffmann E, Fouretier A, Vergne C, Bertram D. Pharmacovigilance regulatory requirements in Latin America. Pharm Med. 2012;26:153–64.

Article  Google Scholar 

Walum E. Acute oral toxicity. Env Health Persp. 1998;106:497–503.

CAS  Google Scholar 

Orellana EA, Kasinski AL. Sulforhodamine B (SRB) assay in cell culture to investigate cell proliferation. Bio-Prot. 2006;6:e1984.

Google Scholar 

Shelanski ML, Gaskin F, Cantor CR. Microtubule assembly in the absence of added nucleotides. Proc Natl Acad Sci. 1973;70:765–68.

Article  CAS  PubMed  PubMed Central  Google Scholar 

Padalia RC, Verma RS, Chauhan A, Goswami P, Singh VR, et al. p-Menthenols chemotype of Cymbopogon distans from India: composition, antibacterial and antifungal activity of the essential oil against pathogens. J Essential Oil Res. 2018;30:40–6.

Article  CAS  Google Scholar 

Nyaa LBT, Tapondjou LA, Barboni L, Tamokou JDD, Kuiate JR, Tane P, et al. NMR assignment and antimicrobial/antioxidant activities of 1β- hydroxyeuscaphic acid from the seeds of Butyrospermum parkii. Nat Prod Sci. 2009;15:76–82.

CAS  Google Scholar 

Septama AW, Panichayupakaranant P. Synergistic effect of artocarpin on antibacterial activity of some antibiotics against methicillin-resistant Staphylococcus aureus, Pseudomonas aeruginosa, and Escherichia coli. Pharm Biol. 2016;54:686–91.

Article  CAS  PubMed  Google Scholar 

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