1. Genick, C. C., Barlier, D., Monna, D. Applications of Biophysics in High-Throughput Screening Hit Validation. J. Biomol. Screen. 2014, 19, 707–714.
Google Scholar | SAGE Journals2. Rainard, J. M., Pandarakalam, G. C., McElroy, S. P. Using Microscale Thermophoresis to Characterize Hits from High-Throughput Screening: A European Lead Factory Perspective. SLAS Discov. 2018, 23, 225–241.
Google Scholar | Abstract3. Coyle, J., Walser, R. Applied Biophysical Methods in Fragment-Based Drug Discovery. SLAS Discov. 2020, 25, 471–490.
Google Scholar | Medline4. Linke, P., Amaning, K., Maschberger, M. An Automated Microscale Thermophoresis Screening Approach for Fragment-Based Lead Discovery. J. Biomol. Screen. 2015, 21, 414–421.
Google Scholar | SAGE Journals5. Seashore-Ludlow, B., Lundbäck, T. Early Perspective: Microplate Applications of the Cellular Thermal Shift Assay (CETSA). J. Biomol. Screen. 2016, 21, 1019–1033.
Google Scholar | SAGE Journals6. Maia de, Oliveira, T., van Beek, L., Shilliday, F. Cryo-EM: The Resolution Revolution and Drug Discovery. SLAS Discov. 2020, 26, 17–31.
Google Scholar | Medline7. Almeida, T., Panova, S., Walser, R. NMR Reporter Assays for the Quantification of Weak Affinity Receptor-Ligand Interactions. SLAS Discov. 2021, 26, 1020–1028.
Google Scholar8. Martinez, W., Arenas, J., Mok, L. Bioelectronic Measurement of Target Engagement to a Membrane-Bound Transporter. SLAS Discov. 2021, 26, 1004–1013.
Google Scholar9. Gradl, S., Steuber, H., Weiske, J. Discovery of the SMYD3 Inhibitor BAY-6035 Using Thermal Shift Assay (TSA) Based High-Throughput Screening. SLAS Discov. 2021, 26, 947–960.
Google Scholar10. Kartal, O., Andres, F., Lai, M. WaveRAPID—A Robust Assay for High-Throughput Kinetic Screens with the Creoptix WAVEsystem. SLAS Discov. 2021, 26, 995–1003.
Google Scholar11. Jeridi, S., Rak, A., Gupta, A. Fast Mek1 Hit Identification with TRIC Technology Correlates Well with Other Biophysical Methods. SLAS Discov. 2021, 26, 1014–1019.
Google Scholar12. Cho, E., Dalby, K. Luminescence Energy Transfer-Based Screening and Target Engagement Approaches for Chemical Biology and Drug Discovery. SLAS Discov. 2021, 26, 984–994.
Google Scholar13. Simon, R., Heabe, T., Ries, R. Acoustic Ejection Mass Spectrometry—A Fully Automatable Technology for High-Throughput Screening in Drug Discovery. SLAS Discov. 2021, 26, 961–973.
Google Scholar14. Scholle, M., McLaughlin, D., Gurard-Levin, Z. High-Throughput Affinity Selection Mass Spectrometry Using SAMDI-MS to Identify Small Molecule Binders of the Human Rhinovirus 3C Protease. SLAS Discov. 2021, 26, 974–983.
Google Scholar