Optimizing Nateglinide Liquisolid Compacts: Achieving Formulation Excellence Through the Quality by Design Approach

Hörter D, Dressman JB. Influence of physicochemical properties on dissolution of drugs in the gastrointestinal tract. Adv Drug Deliv Rev. 2001;46(1–3):75–87.

Article  PubMed  Google Scholar 

Vemula SK, Veerareddy PR. Fast disintegrating tablets of flurbiprofen: formulation and characterization. Lat Am J Pharm. 2011;30(6):1135–41.

CAS  Google Scholar 

Bonthagarala B, Dasari V, Kotra V, Swain S, Beg S. Quality-by-design based development and characterization of pioglitazone loaded liquisolid compact tablets with improved biopharmaceutical attributes. J Drug Deliv Sci Technol. 2019;51:345–55.

Article  CAS  Google Scholar 

Gursoy RN, Benita S. Self-emulsifying drug delivery systems (SEDDS) for improved oral delivery of lipophilic drugs. Biomed Pharmacother. 2004;58(3):173–82.

Article  PubMed  Google Scholar 

Jin X, Zhang Z, Sun E, Li S, Jia X. Statistically designed enzymatic hydrolysis of an icariin/β-cyclodextrin inclusion complex optimized for production of icaritin. Acta Pharm Sin B. 2012;2(1):83–9.

Article  CAS  Google Scholar 

Sonoda R, Horibe M, Oshima T, Iwasaki T, Watano S. Improvement of Dissolution Property of Poorly Water-Soluble drug by Novel Dry Coating Method using Planetary Ball Mill. Chem Pharm Bull (Tokyo). 2008;56(9):1243–7.

Article  CAS  PubMed  Google Scholar 

Blagden N, de Matas M, Gavan PT, York P. Crystal engineering of active pharmaceutical ingredients to improve solubility and dissolution rates. Adv Drug Deliv Rev. 2007;59(7):617–30.

Article  CAS  PubMed  Google Scholar 

Braig V, Konnerth C, Peukert W, Lee G. Enhanced dissolution of naproxen from pure-drug, crystalline nanoparticles: a case study formulated into spray-dried granules and compressed tablets. Int J Pharm. 2019;554:54–60.

Article  CAS  PubMed  Google Scholar 

Daravath B, Tadikonda RR, Vemula SK. Formulation and pharmacokinetics of gelucire solid dispersions of flurbiprofen. Drug Dev Ind Pharm. 2015;41(8):1254–62.

Article  CAS  PubMed  Google Scholar 

Simões MF, Pinto RMA, Simões S. Hot-melt extrusion in the pharmaceutical industry: toward filing a new drug application. Drug Discov Today. 2019;24(9):1749–68.

Article  PubMed  Google Scholar 

Lu M, Xing H, Jiang J, Chen X, Yang T, Wang D, et al. Liquisolid technique and its applications in pharmaceutics. Asian J Pharm Sci. 2017;12(2):115–23.

Article  PubMed  Google Scholar 

Spireas SS, Jarowski CI, Rohera BD. Powdered solution technology: principles and mechanism. Pharm Res. 1992;09(10):1351–8.

Article  CAS  Google Scholar 

Vemula SK, Radhika K. Liquisolid compact technique for improvement of the dissolution rate of flurbiprofen: Formulation and evaluation. J Drug Res Dev. 2015;1(1):2470–1009.

Google Scholar 

Spireas S, Wang T, Grover R. Effect of Powder substrate on the Dissolution properties of Methyclothiazide Liquisolid compacts. Drug Dev Ind Pharm. 1999;25(2):163–8.

Article  CAS  PubMed  Google Scholar 

Javadzadeh Y, Siahi MR, Asnaashari S, Nokhodchi A. An investigation of Physicochemical Properties of Piroxicam Liquisolid Compacts. Pharm Dev Technol. 2007;12(3):337–43.

Article  CAS  PubMed  Google Scholar 

Daravath B, Somalanka S. Enhancement of dissolution rate of racecadotril by liquisolid compact technology. Braz J Pharm Sci. 2022;58:1–14.

Article  Google Scholar 

Javadzadeh Y, Jafari-Navimipour B, Nokhodchi A. Liquisolid technique for dissolution rate enhancement of a high dose water-insoluble drug (carbamazepine). Int J Pharm. 2007;341(1–2):26–34.

Article  CAS  PubMed  Google Scholar 

Spireas S, Sadu S, Grover R. In Vitro Release evaluation of Hydrocortisone Liquisolid tablets. J Pharm Sci. 1998;87(7):867–72.

Article  CAS  PubMed  Google Scholar 

Bhattacharya S, Pasha I, Verma A, Kothapalli R, Jafar F, Hr K. Formulation and evaluation of liquisolid compact of azithromycin dihydrate. J Res Pharm. 2019;23(6):1022–32.

Google Scholar 

Vaskula S, Vemula SK, Bontha VK, Garrepally P. Liquisolid compacts: an approach to enhance the dissolution rate of nimesulide. J Appl Pharm Sci. 2012;2(5):115–21.

Google Scholar 

Chella N, Shastri N, Tadikonda RR. Use of the liquisolid compact technique for improvement of the dissolution rate of valsartan. Acta Pharm Sin B. 2012;2(5):502–8.

Article  Google Scholar 

Swain S, Parhi R, Jena BR, Babu SM. Quality by design: Concept to Applications. Curr Drug Discov Technol. 2019;16(3):240–50.

Article  CAS  PubMed  Google Scholar 

Yu LX, Amidon G, Khan MA, Hoag SW, Polli J, Raju GK, et al. Understanding Pharmaceutical Quality by Design. AAPS J. 2014;16(4):771–83.

Article  CAS  PubMed  PubMed Central  Google Scholar 

Vemula SK, Daravath B, Repka M. Quality by design (QbD) approach to develop fast-dissolving tablets using melt-dispersion paired with surface-adsorption method: formulation and pharmacokinetics of flurbiprofen melt-dispersion granules. Drug Deliv Transl Res. 2023;13(12):3204–22.

Article  CAS  PubMed  Google Scholar 

Bhupinder Singh Bhoop. Quality by design (QbD) for Holistic Pharma Excellence and Regulatory Compliance. Pharma Times. 2014;46(8):26–33.

Google Scholar 

Campbell IW. Nateglinide - current and future role in the treatment of patients with type 2 diabetes mellitus. Int J Clin Pract. 2005;59(10):1218–28.

Article  CAS  PubMed  Google Scholar 

Maggi L, Bruni G, Maietta M, Canobbio A, Cardini A, Conte U. II. Technological approaches to improve the dissolution behavior of nateglinide, a lipophilic insoluble drug: co-milling. Int J Pharm. 2013;454(1):568–72.

Article  CAS  PubMed  Google Scholar 

Okamura A, Emoto A, Koyabu N, Ohtani H, Sawada Y. Transport and uptake of nateglinide in Caco-2 cells and its inhibitory effect on human monocarboxylate transporter MCT1. Br J Pharmacol. 2002;137(3):391–9.

Article  CAS  PubMed  PubMed Central  Google Scholar 

Mamatha T, Sultana N. Enhancement of the dissolution rate of nateglinide tablets using liquisolid compact technique. Asian J Pharm Clin Res. 2017;10(10):241–7.

Article  CAS  Google Scholar 

Daravath B, Naveen C, Vemula SK, Tadikonda RR. Solubility and dissolution enhancement of flurbiprofen by solid dispersion using hydrophilic carriers. Braz J Pharm Sci. 2018;53(4):1–10.

Article  Google Scholar 

Jaydip B, Dhaval M, Soniwala MM, Chavda J. Formulation and optimization of liquisolid compact for enhancing dissolution properties of efavirenz by using DoE approach. Saudi Pharm J. 2020;28(6):737–45.

Article  CAS  PubMed  PubMed Central  Google Scholar 

Elkordy AA, Tan XN, Essa EA. Spironolactone release from liquisolid formulations prepared with Capryol™ 90, Solutol® HS-15 and Kollicoat® SR 30 D as non-volatile liquid vehicles. Eur J Pharm Biopharm. 2013;83(2):203–23.

Article  CAS  PubMed  Google Scholar 

Tayel SA, Soliman II, Louis D. Improvement of dissolution properties of carbamazepine through application of the liquisolid tablet technique. Eur J Pharm Biopharm. 2008;69(1):342–7.

Article  CAS  PubMed  Google Scholar 

Daravath B, Rao Tadikonda R. Formulation and evaluation of meclizine hydrochloride fast dissolving tablets using solid dispersion method. Asian J Pharm Clin Res. 2014;7(2):98–102.

Google Scholar 

Chella N, Daravath B, Kumar D, Tadikonda RR. Formulation and pharmacokinetic evaluation of Polymeric dispersions Containing Valsartan. Eur J Drug Metab Pharmacokinet. 2016;41(5):517–26.

Article  CAS  PubMed  Google Scholar 

Daravath B. Surface solid dispersion: a novel method for improving in-vitro dissolution and in-vivo

留言 (0)

沒有登入
gif