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Alzheimer's disease
Butylcholinesterase inhibitors
Combinatorial chemistry
Conformational restriction
Microscale synthesis
AbbreviationsBuChEbutyrylcholinesterase
PASperipheral anionic site
CuAACCopper-catalysed azide–alkyne cycloadditions
Cdc25Cell division cycle 25
HIVhuman immunodeficiency virus
HATU2-(7-aza-1H-benzotriazole-1-yl)-1,1,3,3-tetramethyluronium hexafluorophosphate
EDC·HCl1-(3-Dimethylaminopropyl)-3-ethylcarbodiimide hydrochloride
TLCthin-layer chromatography
APPamyloid precursor protein
CNScentral nervous system
PAMPAparallel artificial membrane permeability assay
Data availabilityData will be made available on request.
© 2023 Elsevier Inc. All rights reserved.
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