Trans-eyelid distribution of epinastine to the conjunctiva following eyelid application in rabbits

Leonardi A, Motterle L, Bortolotti M. Allergy and the eye. Clin Exp Immunol. 2008;153(suppl 1):17–21.

Article  CAS  PubMed  PubMed Central  Google Scholar 

Abelson MB, Shetty S, Korchak M, Butrus SI, Smith LM. Advances in pharmacotherapy for allergic conjunctivitis. Expert Opin Pharmacother. 2015;16:1219–31.

Article  CAS  PubMed  Google Scholar 

Chrai SS, Patton TF, Mehta A, Robinson JR. Lacrimal and instilled fluid dynamics in rabbit eyes. J Pharm Sci. 1973;62:1112–21.

Article  CAS  PubMed  Google Scholar 

Pahuja P, Arora S, Pawar P. Ocular drug delivery system: a reference to natural polymers. Expert Opin Drug Deliv. 2012;9:837–61.

Article  CAS  PubMed  Google Scholar 

Leonardi A, Silva D, Formigo DP, Bozkurt B, Sharma V, Allegri P, et al. Management of ocular allergy. Allergy. 2019;74:1611–30.

Article  PubMed  Google Scholar 

Miyazaki D, Takamura E, Uchio E, Ebihara N, Ohno S, Ohashi Y, et al. Japanese guidelines for allergic conjunctival diseases 2020. Allergol Int. 2020;69:346–55.

Article  CAS  PubMed  Google Scholar 

Dupuis P, Prokopich CL, Hynes A, Kim H. A contemporary look at allergic conjunctivitis. Allergy Asthma Clin Immunol. 2020;16:5.

Article  PubMed  PubMed Central  Google Scholar 

Vogelson CT, Abelson MB, Pasquine T, Stephens DM, Gamache DA, Gross RD, et al. Preclinical and clinical antiallergic effect of olopatadine 0.2% solution 24 hours after topical ocular administration. Allergy Asthma Proc. 2004;25:69–75.

CAS  PubMed  Google Scholar 

Torkildsen G, Narvekar A, Bergmann M. Efficacy and safety of olopatadine hydrochloride 0.77% in patients with allergic conjunctivitis using a conjunctival allergen-challenge model. Clin Ophthalmol. 2015;9:1703–13.

Article  CAS  PubMed  PubMed Central  Google Scholar 

McLaurin E, Narvekar A, Gomes P, Adewale A, Torkildsen G. Phase 3 randomized double-masked study of efficacy and safety of once-daily 0.77% olopatadine hydrochloride ophthalmic solution in subjects with allergic conjunctivitis using the conjunctival allergen challenge model. Cornea. 2015;34:1245–51.

Article  PubMed  Google Scholar 

Greiner JV, Edwards-Swanson K, Ingerman A. Evaluation of alcaftadine 0.25% ophthalmic solution in acute allergic conjunctivitis at 15 minutes and 16 hours after instillation versus placebo and olopatadine 0.1%. Clin Ophthalmol. 2011;5:87–93.

CAS  PubMed  PubMed Central  Google Scholar 

Gote V, Sikder S, Sicotte J, Pal D. Ocular drug delivery: present innovations and future challenges. J Pharmacol Exp Ther. 2019;370:602–24.

Article  CAS  PubMed  Google Scholar 

Jumelle C, Gholizadeh S, Annabi N, Dana R. Advances and limitations of drug delivery systems formulated as eye drops. J Control Release. 2020;321:1–22.

Article  CAS  PubMed  PubMed Central  Google Scholar 

Abdi B, Mofidfar M, Hassanpour F, Cilingir EK, Kalajahi SK, Milani PH, et al. Therapeutic contact lenses for the treatment of corneal and ocular surface diseases: advances in extended and targeted drug delivery. Int J Pharm. 2023;638:122740.

Article  CAS  PubMed  Google Scholar 

Kimura C, Tojo K. Development of a stick-type transdermal eyelid delivery system of ketotifen fumarate for ophthalmic diseases. Chem Pharm Bull. 2007;55:1002–5.

Article  CAS  Google Scholar 

See GL, Arce F Jr, Itakura S, Todo H, Sugibayashi K. Prolonged distribution of tranilast in the eyes after topical application onto eyelid skin. Chem Pharm Bull. 2020;68:779–83.

Article  CAS  Google Scholar 

Ogura N, Fujisawa K, Kato M. Epinastine cream: a novel once-daily therapeutic agent for allergic conjunctivitis. J Ocul Pharmacol Ther. 2024;40:173–80.

Article  CAS  PubMed  Google Scholar 

Scheuplein RJ. Mechanism of percutaneous absorption. II. Transient diffusion and the relative importance of various routes of skin penetration. J Invest Dermatol. 1967;48:79–88.

Article  CAS  PubMed  Google Scholar 

Vickers CF. Existence of reservoir in the stratum corneum. Experimental Proof Arch Dermatol. 1963;88:20–3.

Article  CAS  PubMed  Google Scholar 

Tse S, Powell KD, Maclennan SJ, Moorman AR, Paterson C, Bell RR. Skin permeability and pharmacokinetics of diclofenac epolamine administration by dermal patch in Yorkshire-Landrace pigs. J Pain Res. 2012;5:401–8.

Article  CAS  PubMed  PubMed Central  Google Scholar 

van den Heuvel MW, van Bragt AJM, Alnabawy AKM, Kaptein MCJ. Comparison of ethinylestradiol pharmacokinetics in three hormonal contraceptive formulations: the vaginal ring, the transdermal patch and an oral contraceptive. Contraception. 2005;72:168–74.

Article  PubMed  Google Scholar 

Pratchyapruit W, Kikuchi K, Gritiyarangasan P, Aiba S, Tagami H. Functional analyses of the eyelid skin constituting the most soft and smooth area on the face: contribution of its remarkably large superficial corneocytes to effective water-holding capacity of the stratum corneum. Skin Res Technol. 2007;13:169–75.

Article  PubMed  Google Scholar 

Ya-Xian Z, Suetake T, Tagami H. Number of cell layers of the stratum corneum in normal skin – relationship to the anatomical location on the body, age, sex and physical parameters. Arch Dermatol Res. 1999;291:555–9.

Article  CAS  PubMed  Google Scholar 

Nicolau PJ. The orbicularis oris muscle: a functional approach to its repair in the cleft lip. Br J Plast Surg. 1983;36:141–53.

Article  CAS  PubMed  Google Scholar 

Most SP, Mobley SR, Larrabee WF Jr. Anatomy of the eyelids. Facial Plast Surg Clin North Am. 2005;13:487–92.

Article  PubMed  Google Scholar 

Beard C. Muller’s superior tarsal muscle: anatomy, physiology, and clinical significance. Ann Plast Surg. 1985;14:324–33.

Article  CAS  PubMed  Google Scholar 

Cahill JF, Kertesz V, Weiskittel TM, Vavrek M, Freddo C, van Berkel GJ. Online, absolute quantitation of propranolol from spatially distinct 20- and 40-µm dissections of brain, liver, and kidney thin tissue sections by laser microdissection-liquid vortex capture-mass spectrometry. Anal Chem. 2016;88:6026–34.

Article  CAS  PubMed  Google Scholar 

Hollingshead BD, Tomlinson L, Finley J, Doshna C, Ritenour C, Barricklow J, et al. An orthogonal methods assessment of topical drug concentrations in skin and the impact for risk assessment in the viable epidermis. Regul Toxicol Phrmacol. 2021;123:104934.

Article  CAS  Google Scholar 

Kaya F, Zimmerman MD, Antilus-Sainte R, Gengenbacher M, Carter CL, Dartois V. Spatial quantitation of antibiotics in bone tissue compartments by laser-capture microdissection coupled with UHPLC-tandem mass spectrometry. Anal Bioanal Chem. 2022;414:6919–27.

Article  CAS  PubMed  PubMed Central  Google Scholar 

Mori N, Mochizuki T, Yamazaki F, Takei S, Mano H, Matsugi T, et al. MALDI imaging mass spectrometry revealed atropine distribution in the ocular tissues and its transit from anterior to posterior regions in the whole-eye of rabbit after topical administration. PLoS ONE. 2019;14:e0211376.

Article  CAS  PubMed  PubMed Central  Google Scholar 

Bonnel D, Legouffe R, Eriksson AH, Mortensen RW, Pamelard F, Stauber J, et al. MALDI imaging facilitates new topical drug development process by determining quantitative skin distribution profiles. Anal Bioanal Chem. 2018;410:2815–28.

Article  CAS  PubMed  Google Scholar 

Solon EG. Use of radioactive compounds and autoradiography to determine drug tissue distribution. Chem Res Toxicol. 2012;25:543–55.

Article  CAS  PubMed  Google Scholar 

Solon EG, Schweitzer A, Stoeckli M, Prideaux B, Autoradiography. MALDI-MS, and SIMS-MS imaging in pharmaceutical discovery and development. AAPS J. 2010;12:11–26.

Article  CAS  PubMed  Google Scholar 

Prideaux B, Lenaerts A, Dartois V. Imaging and spatially resolved quantification of drug distribution in tissues by mass spectrometry. Curr Opin Chem Biol. 2018;44:93–100.

Article  CAS  PubMed  Google Scholar 

Ikeda H, Sato M, Tsukamoto H, Sato E, Unei H, Kimura Y, et al. Evaluation and multivariate statistical analysis of factors influencing patient adherence to ophthalmic solutions. Yakugaku Zasshi. 2001;121:799–806.

Article  CAS  PubMed  Google Scholar 

Tsumura T, Kashiwagi K, Suzuki Y, Yoshikawa K, Suzumura H, Maeda T, et al. A nationwide survey of factors influencing adherence to ocular hypotensive eyedrops in Japan. Int Ophthalmol. 2019;39:375–83.

Article  PubMed  Google Scholar 

Gurwitz JH, Glynn RJ, Monane M, Everitt DE, Gilden D, Smith N, et al. Treatment for glaucoma: adherence by the elderly. Am J Public Health. 1993;83:711–6.

留言 (0)

沒有登入
gif